Cat. No. |
Product Name |
Information |
PC-72602 |
Cotadutide acetate
Dual GLP-1/glucagon receptor agonist
|
Cotadutide acetate (MEDI-0382, MEDI0382) is a potent dual GLP-1/glucagon receptor peptide agonist with EC50 values of 6.9 pM and 10.2 pM, respectively. |
PC-20600 |
RGT1383
GLP-1R agonist
|
RGT1383 is a small molecule GLP-1R agonist, RGT1383 is a full agonist in G protein-mediated cAMP signaling with EC50 of 0.2 nM, and a partial agonist in β-arrestin-mediated signaling. |
PC-20512 |
LSN3318839
GLP-1R PAM
|
LSN3318839 is a potent, positive allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R) with EC50 of 14 nM, Emax of 104%. |
PC-72853 |
V-0219
GLP-1R PAM
|
V-0219 is a small molecule positive allosteric modulator (PAM) of GLP-1R with Emax of 60% in the cAMP assay. |
PC-72213 |
TT-OAD2 hydrochloride
GLP-1 agonist
|
TT-OAD2 hydrochloride is a potent, selective, non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor with EC50 of 5 nM. |
PC-72212 |
TT-OAD2
GLP-1 agonist
|
TT-OAD2 is a potent, selective, non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor with EC50 of 5 nM. |
PC-72210 |
Danuglipron
GLP-1 agonist
|
Danuglipron (PF-06882961) is a potent, selective, non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor. |
PC-35834 |
NLY01
|
NLY01 (NLY-01, GLP1R agonist NLY01) is a potent, brain-penetrant long-acting GLP1R agonist, protects against the loss of dopaminergic neurons and behavioral deficits in the α-synuclein preformed fibril (α-syn PFF) mouse model of sporadic Parkinson's disease, blocks the microglial activation and the generation of A1 astrocytes. |
PC-43539 |
Exenatide acetate
|
Exenatide acetate (Exendin-4 acetate) is the acetate of Exenatide, which is highly potent, long-acting glucagon-like peptide-1 receptor (GLP-1) agonist with IC50 of 3.22 nM.. |
PC-43093 |
LGD-6972
|
LGD-6972 (RVT 1502) is a novel potent, selective, orally bioavailable glucagon receptor (GCGR) antagonist. |
PC-61363 |
Apraglutide
|
A peptidic glucagon like peptide 2 (GLP-2) analogue for treatment of type2 diabetes.. |
PC-70259 |
GLP1-agonist-1
|
A potent, selective GLP-1 agonist. |