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Cat. No. Product Name Information
PC-38112

BMS-820132

BMS-820132 (BMS 820132) is potent, selective, partial glucokinase (GK) activator with AC50 of 29 nM.
PC-36020

TTP399

GK activator

Cadisegliatin (TTP399) is a hepatoselective, oral Glucokinase (GK) activator with EC50 of 304 nM and 762 nM for human GK at high glucose concentration (15 mM) and normoglycemia (5 mM), respectively.
PC-61879

MK-0941 mesylate

MK-0941 mesylate (MK0941) is a novel potent, orally active Glucokinase (GK) activator with EC50 of 0.240 and 0.065 uM in 2.5 and 10 mM glucose, respectively.
PC-61878

MK-0941

MK-0941 (MK0941) is a novel potent, orally active Glucokinase (GK) activator with EC50 of 0.240 and 0.065 uM in 2.5 and 10 mM glucose, respectively.
PC-60040

Dorzagliatin

Dorzagliatin (HMS-5552, HMS5552) is a novel potent, fourth-generation glucokinase (GK) activator.
PC-42091

AM-2394

Glucokinase activator

A potent, orally bioavailable Glucokinase (GK) activator with EC50 of 60 nM.
PC-49838

TMG-123

Glucokinase activator

TMG-123 (TMG123) is a potent small molecule activator of glucokinase (GK) with EC50 of 0.35 and 0.32 uM for human liver and pancreas GK, respectively.
PC-49837

GKM-001

Glucokinase activator

GKM-001 is a potent, liver-selective small molecule activator of glucokinase (GKA), demonstrates glucose lowering effect without hypoglycemia in normal and type II diabetes mellitus (T2DM).
PC-49836

LY2608204

Glucokinase activator

Globalagliatin (LY2608204) is a potent, small molecule activator of glucokinase (GK) with EC50 value of 42 nM, induces glucose metabolism and reduces glucose levels for the treatment of type 2 diabetes.
PC-49835

PF-04937319

Glucokinase activator

PF-04937319 (PB-201, PF 4937319) is a partial, pancreas/liver-dual glucokinase activator with EC50 of 174 nM, induces glucose metabolism and reduces glucose levels for the treatment of type 2 diabetes.
PC-49834

AMG 151

Glucokinase activator

AMG 151 (ARRY-403) is an orally available allosteric glucokinase activator developed for the treatment of diabetes.
PC-49828

GKA23

Glucokinase activator

GKA23 is a potent, small molecule glucokinase (GK) activator with EC50 of 152 nM for glucokinase activation in 5 mM glucose, increases glucose uptake in primary rat hepatocytes with EC50 of 201 nM.

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