Histamine Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-23506	Latrepirdine 3613-73-8	Latrepirdine (Dimebolin, Dimebone) is a neuroactive compound with antagonist activity at histaminergic, α-adrenergic, and serotonergic receptors, stimulates amyloid precursor protein (APP) catabolism and amyloid-β (Aβ) secretion.
PC-23486	Ketotifen PDE8B inhibitor	Ketotifen (HC 20-511) is an orally active second-generation noncompetitive histamine 1 (H1) receptor blocker and mast cell stabilizer, also is a PDE8B inhibitor.
PC-23473	JNJ-7777120 H4R antagonist	JNJ-7777120 (JNJ 7777120) is potent and selective histamine H4 receptor (H4R) antagonist with Ki of 4.5 nM (hH4R), >1000-fold selectivity over H1, H2, or H3 receptors.
PC-23262	Izuforant H4R antagonist	Izuforant (JW1601, LEO 152020) is a potent, selective and oral histamine 4 receptor (H4R) antagonist with IC50 of 65.1-72.2 nM in human whole-blood assay, and pKi of 6.83 and 5.36 at mouse and rat histamine receptor subtypes. shows lower pKi values against other histamine receptor.
PC-42910	Pitolisant oxalate	A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM.

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