| Cat. No. |
Product Name |
Information |
| PC-62976 |
GR-73632
|
GR-73632 is a potent and selective tachykinin NK1 receptor agonist with EC50 of 2 nM, promotes differentiation but not survival of rat chromaffin cells in vitro.. |
| PC-61581 |
Casopitant mesylate
|
Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities. |
| PC-61580 |
Casopitant
|
Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities. |
| PC-61579 |
Vestipitant mesylate
|
Vestipitant (GW597599) is a potent, selective, orally active NK1 receptor antagonist with pKi of 9.65. |
| PC-61578 |
Vestipitant
|
Vestipitant (GW597599) is a potent, selective, orally active NK1 receptor antagonist with pKi of 9.65. |
| PC-61552 |
Orvepitant
|
Orvepitant (GW823296) is a potent and selective, brain penetrant NK1 receptor antagonist with pKi of 10.2. |
| PC-60342 |
SR 140333
|
A potent, selective, non-peptide NK1 receptor antagonist with Ki of 0.74 nM, IC50 of 1.6 nM. |
| PC-60341 |
L-732138
|
A potent, selective and competitive NK1 receptor antagonist with IC50 of 2.3 nM. |
| PC-70194 |
L-733060 hydrochloride
|
An orally active, non-peptide, selective antagonist for the NK1 receptor with Ki of 0.8 nM. |
| PC-70193 |
L-733060
|
An orally active, non-peptide, selective antagonist for the NK1 receptor with Ki of 0.8 nM. |
| PC-70192 |
GR-159897
|
A potent non-peptide antagonist of tachykinin NK2 receptor with pKi of 9.5 in CHO cells. |
| PC-70191 |
Ibodutant
|
A potent and selective linear tachykinin NK2 receptor antagonist with pKb of 9.3. |
