| Cat. No. |
Product Name |
Information |
| PC-60457 |
AZD2716
|
AZD2716(AZD-2716) is a novel potent, selective, orally bioavailable sPLA2 inhibitor with excellent plasma sPLA2 inhibition (IC50=0.1 nM). |
| PC-70212 |
Rilapladib
|
Rilapladib (SB-659032, SB659032) is a potent, selective and oral lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with IC50 of 0.23 nM, for the treatment of Alzheimer's disease and atherosclerosis.. |
| PC-42634 |
Darapladib
|
Darapladib (SB480848) is a potent Lp-PLA2 inhibitor with IC50 of 0.25 nM, shows an enhanced in vitro and in vivo profile versus SB-435495. |
| PC-42702 |
CAY10650
cPLA2α inhibitor
|
CAY10650 is a highly potent cytosolic phospholipase A2α (cPLA2α) inhibitor with an IC50 of 12 nM. |
| PC-22189 |
AX048
cPLA2 inhibitor
|
AX048 is a potent cytosolic group IVA phospholipase A2 (cPLA2) with analgesic effect. |
| PC-20922 |
VU533
NAPE-PLD activator
|
VU533 is a small molecule activator of N-acyl-phosphatidylethanolamine hydrolyzing phospholipase D (NAPE-PLD) with EC50 of 0.3 uM, enhances efferocytosis by macrophages. |
| PC-20921 |
VU534
NAPE-PLD activator
|
VU534 is a small molecule activator of N-acyl-phosphatidylethanolamine hydrolyzing phospholipase D (NAPE-PLD) with EC50 of 0.3 uM, enhances efferocytosis by macrophages. |
| PC-20134 |
ABHD6 inhibitor 22f
ABHD6 inhibitor
|
ABHD6 inhibitor 22f is a potent, selective ABHD6 inhibitor with IC50 of 8.0 nM (hABHD6), does not inhibit hMGL and hFAAH. |
| PC-20133 |
KT-203
ABHD6 inhibitor
|
KT-203 (KT203) is a potent, selective inhibitor of α/β-hydrolase domain 6 (ABHD6) with IC50 of 3.9 nM in 2-AG hydrolysis assays. |
| PC-20132 |
WWL-70
ABHD6 inhibitor
|
WWL-70 is a potent selective inhibitor of α/β-hydrolase domain 6 (ABHD6) with IC50 of 70 nM. |
| PC-20131 |
KT-185
ABHD6 inhibitor
|
KT-185 (KT185) is a potent, selective, irreversible and orally-active α/β-hydrolase domain 6 (ABHD6) inhibitor with IC50 of 0.21 nM. |
| PC-20130 |
KT-182
ABHD6 inhibitor
|
KT-182 (KT182) is a potent, selective, irreversible α/β-hydrolase domain 6 (ABHD6) inhibitor with IC50 of 1.7 nM. |
