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Cat. No. Product Name Information
PC-60963

PR-924

A potent, specific immunoproteasome LMP7 subunit inhibitor with IC50 of 25 nM, >100-fold selectivity over β5c, β1i, β1c, β2i and β2c subunits (IC50>3 uM).
PC-60476

FV-162

A potent, orally bioavailable, irreversible proteasome inhibitor with potent antimyeloma activity (IC50<60 nM).
PC-42596

MLN2238

A potent, selective, orally bioavailable proteasome inhibitor with IC50 of 3.4 nM.
PC-45704

PD-151746

A potent, selective, cell-permeable Calpain inhibitor with Ki of 0.26 uM for m-calpain.
PC-42597

Delanzomib

A potent, orally active proteasome inhibitor with IC50 of 3.8 nM against chymotrypsin-like proteasome activity.
PC-45547

VR-23

A potent inhibitor of trypsin-like proteasome (IC50=1 nM), chymotrypsin-like proteasome (IC50=50-100 nM) and caspase-like proteasome (IC50=3 uM).
PC-45577

MG-101

A potent inhibitor of cysteine proteases including calpain I (Ki= 190 nM), calpain II (Ki= 220 nM), cathepsin B (Ki= 150 nM) and cathepsin L (Ki= 500 pM).
PC-42190

PD-150606

A potent and selective calpain inhibitor with Ki of 0.21 uM/0.37 uM for u-calpain/m-calpain, respectively.

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