| Cat. No. |
Product Name |
Information |
| PC-63070 |
BD-1047
Sigma 1 receptor antagonist
|
BD-1047 is a potent, selecitve Sigma 1 receptor (σ1) antagonist with Ki of 0.93 nM. |
| PC-62827 |
Sigma1-IN-4
Sigma 1 inhibitor
|
Sigma1-IN-4 is a novel small molecule sigma-1 receptor inhibitor with Ki of 38 nM. |
| PC-62223 |
Finazine
Sigma receptor ligand
|
Finazine is a high-affinity, brain penetrant sigma-1 and sigma 2 receptor ligand with Ki of 2.6 nM and 46 nM, respectively. |
| PC-61602 |
4-BBPB
Sigma 1 receptor agonist
|
4-BBPB is a highly potent agonist of sigma 1 receptor (σ1 receptor) with Ki of 0.8 nM. |
| PC-61601 |
4-BBPB maleate
Sigma 1 receptor agonist
|
4-BBPB maleate is a highly potent agonist of sigma 1 receptor (σ1 receptor) with Ki of 0.8 nM. |
| PC-61105 |
MIN-101
5-HT2A/Sigma 2 inhibitor
|
MIN-101 (Roluperidone, CYR-101, MT-210) is a higly potent 5-HT2A and sigma 2 receptor antagonist, with no direct dopamine affinities, for treatment of negative symptoms in schizophrenia.. |
| PC-61104 |
UKH-1114
Sigma 2 receptor agonist
|
UKH-1114 (UKH1114) is a potent, sigma 2 receptor/Tmem97 agonist with Ki of 46 nM. |
| PC-61103 |
SAS-1121
Sigma 2 Receptor ligand
|
SAS-1121 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 16.2 nM, 574-fold selectivity over sigma 1 receptors. |
| PC-61102 |
DKR-1051
Sigma 2 Receptor ligand
|
DKR-1051 is a novel potent, subtype-selective sigma 2 receptor/PGRMC1 ligand with Ki of 61 nM, 9-fold selectivity over sigma 1 receptors (Ki=556 nM). |
| PC-61101 |
JVW-1009
Sigma receptor ligand
|
A small molecule sigma receptor ligand with Ki of 96 and 70 nM for sigma 1 and sigma 2, respectively. |
| PC-61100 |
SAS-0132
Sigma 2 Receptor ligand
|
SAS-0132 (SAS132) is a novel potent, subtype-selective, brain penetrant sigma 2 receptor/PGRMC1 ligand with Ki of 90 nM, 9-fold selectivity over sigma 1 receptors. |
| PC-60790 |
PD144418
Sigma 1 inhibitor
|
PD144418 is a potent, selective sigma 1 ligand with Ki of 0.08 nM, >3000-fold selectivity over sigma 2 (Ki=1377 nM). |
