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Cat. No. Product Name Information
PC-45237

Guanfacine hydrochloride

α2 adrenoceptor agonist

Guanfacine hydrochloride is a selective α2A receptor agonist that can reduce peripheral sympathetic outflow and thus cansues a reduction in peripheral sympathetic tone.
PC-43903

Olodaterol

β2 adrenoceptor agonist

Olodaterol (BI 1744) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2.
PC-45155

Medetomidine

α2-adrenoceptor agonist

Medetomidine is a potent, highly selective α2-adrenoceptor agonist with Ki of 1.08 nM.
PC-42334

Asenapine

5-HT antagonist

Asenapine (Org5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors.
PC-45299

Bambuterol hydrochloride

Bambuterol hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma.
PC-45298

Bambuterol

beta-adrenoceptor agonist

Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline.
PC-42338

Silodosin

α1A-adrenoceptor antagonist

Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM.
PC-22867

AGN-762

α2B/α2C adrenergic receptor activator

AGN-762 is a selective activator of α2B- and α2C-adrenergic receptor subtypes, but not the α2A subtype.
PC-22600

WB4101

α1A adrenoceptor antagonist

WB4101 is a potent, α1A-adrenergic selective antagonist with pKB value of 8.9 in rabbit aorta.
PC-22446

ATR-127

β2/β3-adrenoceptor agonist

ATR-127 is a highly effective β2- and β3-adrenoceptors (ARs) agonist with pEC50 of 6.53 and 5.5 for rat β2-AR and mouse β3-AR, respectively.
PC-22239

SR59230A

β3AR antagonist

SR59230A is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50 of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively.
PC-21223

ZD7114

beta-adrenoceptor agonist

ZD7114 (ICI D7114) is a potent, selective beta-adrenoceptor agonist, selectively stimulates brown fat and increases whole-body oxygen consumption.

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