| Cat. No. |
Product Name |
Information |
| PC-45237 |
Guanfacine hydrochloride
α2 adrenoceptor agonist
|
Guanfacine hydrochloride is a selective α2A receptor agonist that can reduce peripheral sympathetic outflow and thus cansues a reduction in peripheral sympathetic tone. |
| PC-43903 |
Olodaterol
β2 adrenoceptor agonist
|
Olodaterol (BI 1744) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
| PC-45155 |
Medetomidine
α2-adrenoceptor agonist
|
Medetomidine is a potent, highly selective α2-adrenoceptor agonist with Ki of 1.08 nM. |
| PC-42334 |
Asenapine
5-HT antagonist
|
Asenapine (Org5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors. |
| PC-45299 |
Bambuterol hydrochloride
|
Bambuterol hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma. |
| PC-45298 |
Bambuterol
beta-adrenoceptor agonist
|
Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline. |
| PC-42338 |
Silodosin
α1A-adrenoceptor antagonist
|
Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM. |
| PC-22867 |
AGN-762
α2B/α2C adrenergic receptor activator
|
AGN-762 is a selective activator of α2B- and α2C-adrenergic receptor subtypes, but not the α2A subtype. |
| PC-22600 |
WB4101
α1A adrenoceptor antagonist
|
WB4101 is a potent, α1A-adrenergic selective antagonist with pKB value of 8.9 in rabbit aorta. |
| PC-22446 |
ATR-127
β2/β3-adrenoceptor agonist
|
ATR-127 is a highly effective β2- and β3-adrenoceptors (ARs) agonist with pEC50 of 6.53 and 5.5 for rat β2-AR and mouse β3-AR, respectively. |
| PC-22239 |
SR59230A
β3AR antagonist
|
SR59230A is a potent, selective, and blood-brain barrier penetrating β3-adrenergic receptor antagonist with IC50 of 40, 408, and 648 nM for β3, β1, and β2 receptors, respectively. |
| PC-21223 |
ZD7114
beta-adrenoceptor agonist
|
ZD7114 (ICI D7114) is a potent, selective beta-adrenoceptor agonist, selectively stimulates brown fat and increases whole-body oxygen consumption. |
