| Cat. No. |
Product Name |
Information |
| PC-21196 |
Mirabegron
β3-adrenoceptor agonist
|
Mirabegron (YM178) is a potent, selective selective β3-adrenoceptor agonist with EC50 of 22.4 nM. |
| PC-20987 |
Difluorophenyl Quinazoline
β2AR modulator
|
Difluorophenyl Quinazoline (DFPQ, AP-06-202) is a selective, biased, negative allosteric modulator of β-arrestin recruitment to the β2AR, without effect on on β2AR coupling to Gs. |
| PC-20986 |
L-771688
α1A adrenoceptor antagonist
|
L-771688 (L-771,688, SNAP 6383) is a potent and selective alpha1A (α1A)-adrenoceptor antagonist with binding Ki of 0.13 nM to α1-adrenoceptors in human prostate tissue. |
| PC-20804 |
Nebivolol hydrochloride
Beta adrenergic antagonist
|
Nebivolol hydrochloride (R 065824) is a beta adrenergic antagonist and shows direct vasodilator properties and adrenergic blocking characteristics. |
| PC-43177 |
Midodrine hydrochloride
|
Midodrine is a selective α1-adrenoceptor agonist that acts as a vasopressor/antihypotensive agent for the treatment of dysautonomia and orthostatic hypotension. |
| PC-43176 |
Midodrine
|
Midodrine is a selective α1-adrenoceptor agonist that acts as a vasopressor/antihypotensive agent for the treatment of dysautonomia and orthostatic hypotension. |
| PC-43161 |
Yohimbine
|
Yohimbine is an indole alkaloid that has high affinity for the α2-adrenergic receptors with Ki of 1 nM for α2A, α2B and α2C. |
| PC-43012 |
Atipamezole
|
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM. |
| PC-43011 |
Atipamezole hydrochloride
|
Antipamezole (MPV-1248) is a potent, specific α2-adrenoceptor antagonist with Ki of 1.6 nM. |
| PC-42808 |
Asenapine maleate
|
Asenapine maleate (Org 5222) is a potent psychopharmacologic agent that shows high affinity for 5-HT, dopamine, histamine and adrenoceptors. |
| PC-62005 |
Milveterol hydrochloride
|
Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold). |
| PC-62004 |
Milveterol
|
Milveterol (GSK 159797) is a potent, selective long-acting β2 adrenoceptor agonist with pEC50 of 10.2 in cell-based assays, displays good β2/β1 selectivity (>300-fold). |
