| Cat. No. |
Product Name |
Information |
| PC-45155 |
Medetomidine
α2-adrenoceptor agonist
|
Medetomidine is a potent, highly selective α2-adrenoceptor agonist with Ki of 1.08 nM. |
| PC-45270 |
Salmeterol
β2AR agonist
|
Salmeterol (GR33343X) is a long-acting beta2-adrenergic receptor agonist (Ki=1.5 nM) used clinically to treat asthma and maintenance of COPD. |
| PC-45299 |
Bambuterol hydrochloride
|
Bambuterol hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma. |
| PC-45298 |
Bambuterol
beta-adrenoceptor agonist
|
Bambuterol is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; also is a prodrug of terbutaline. |
| PC-42338 |
Silodosin
α1A-adrenoceptor antagonist
|
Silodosin (KAD3213, KMD3213) is a highly potent, uroselective α1a-adrenoceptor antagonist with Ki of 36 pM. |
| PC-26836 |
Terazosin
PGK1 activator, α1-adrenergic receptor antagonist
|
Terazosin is a small molecule α1-adrenergic receptor antagonist and activator of phosphoglycerate kinase 1 (PGK1) at 2.5 nM -0.5 uM, binds to PGK1 with ITC Kd of 2.78 uM. |
| PC-26658 |
RX821002
α2A/D-adrenoreceptor antagonist
|
RX821002 (2-Methoxyidazoxan) is a highly selective antagonist of alpha2A/D-adrenoreceptor (alpha2A/D-AR) antagonist with pKd of 8.2 and 9.7 for rabbit alpha 2A-adrenoceptor and guinea-pig alpha 2D-adrenoceptor respectively. |
| PC-26581 |
A-61603
α1A AR agonist
|
A-61603 is a potent, selective alpha 1-adrenergic receptor (α1A AR) agonist, >35-fold more potent at α1A than at α1B or α1D sites, induces dose response increases in spontaneous Ca2+ transients in rat ventricular myocytes in vitro with EC50 of 6.9 nM. |
| PC-25621 |
Trifluoperazine
eEF2K inhibitor, α1-adrenergic receptor antagonist
|
Trifluoperazine is an antiadrenergic, antidopaminergic and anticholinergic agent, potent α1-adrenergic receptor antagonist, also inhibits calcium/calmodulin to eEF2K. |
| PC-25616 |
Vatinoxan hydrochloride
α2A adrenoceptor antagonist
|
Vatinoxan hydrochloride (MK-467, L-659066) is a potent and selective alpha-2 adrenoceptor (α2A adrenoceptor, α2AR) antagonist with IC50 of 3 nM against the binding of [3H]rauwolscine to rat cerebrocortical membranes, selective over alpha-1 adrenoceptors. |
| PC-25423 |
Formoterol fumarate
β2-adrenoceptor agonist
|
Formoterol fumarate is a potent, selective and long-acting β2-adrenoceptor agonist. |
| PC-25233 |
Imiloxan hydrochloride
α2B adrenoceptor antagonist
|
Imiloxan hydrochloride (RS 21361) is a potent and selective alpha 2B-adrenoceptor antagonist. |
