| Cat. No. |
Product Name |
Information |
| PC-35866 |
IMTPPE
AR inhibitor
|
IMTPPE (SID 3712502) is a novel small molecule capable of inhibiting androgen receptor (AR) transcriptional activity (IC50=1 uM) and protein level in C4-2 prostate cancer cells. |
| PC-35680 |
KCI807
AR-ELK1 inhibitor
|
KCI807 (KCI-807) is a small molecule that selectively disrupts ELK1-dependent promoter activation by wild-type and variant androgen receptors (IC50=0.53 uM) without interfering with ELK1 activation by ERK. |
| PC-35346 |
RD162
AR antagonist
|
RD162 is a second-generation, orally available antiandrogen that binds to androgen receptor (AR) with IC50 of 30.9 nM. |
| PC-35143 |
LGD-2226
SARM
|
LGD-2226 (LGD2226) is an orally active, selective androgen receptor modulator (SARM) with binding Ki of 1 nM, >1000-fold selectivity over GR,PR, MR and ER. |
| PC-35133 |
LY305
SARM
|
LY305 (LY-305) is a non-steroidal selective androgen receptor modulator (SARM) with Ki of 2.03 nM, demonstrates potent agonist activity in the aforementioned C2C12 cellular assay (EC50=0.499 nM). |
| PC-35003 |
BAY 1024767
AR antagonist
|
BAY 1024767 (BAY1024767) is a higly potent antagonist of androgen receptor (AR) wild-type (IC50=46 nM) and mutant forms located in the AR ligand-binding domain (LBD). |
| PC-43500 |
Cortexolone 17 alpha-propionate
Androgen antagonist
|
Cortexolone 17 alpha-propionate (CB-03-01, Clascoterone) is a topical and peripherally selective androgen antagonist, displays a strong local antiandrogenic activity in hamster's flank organ test, does not exhibit antiandrogenic activity after subcutaneous injection in vivo. |
| PC-43002 |
Trenbolone acetate
|
Trenbolone acetate (RU-1697,17beta-TBOH) is a potent testosterone analog and selective androgen receptor modulator, is an androgen ester and a long-acting prodrug of trenbolone. |
| PC-42895 |
BMS-564929
SARM
|
BMS-564929 is a potent, selective androgen receptor modulator (SARM) that binds to AR with Ki of 2.11 nM. |
| PC-42838 |
Andarine
SARM
|
Andarine (S4, GTx007) is a non-steroidal selective androgen receptor modulator (SARM) with Ki of 4 nM, efficaciously stimulates AR-mediated reporter gene expression. |
| PC-62000 |
Ostarine
SARM
|
Ostarine (Enobosarm, GTx-024, MK-2866) is a selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and osteoporosis. |
| PC-61999 |
LY2452473
SARM
|
LY2452473 (TT 701, OPK 88004) is an orally bioavailable selective androgen receptor modulator (SARM) being developed for the treatment of disorders related to hypogonadism. |
