You are here:Home-Chemical Inhibitors & Agonists-Others-CaMK

Request The Product List ofCaMK CaMK

Cat. No. Product Name Information
PC-21443

CC-8977

CaMKK2 inhibitor

CC-8977 is a hgihly potent, selective inhibitor of calcium/calmodulin-dependent kinase kinase II (CaMKK2) with binding IC50 of 7 nM.
PC-49624

SGC-CAMKK2-1N

SGC-CAMKK2-1N is the negative control compound of the CaMKK2 inhibitor SGC-CAMKK2-1 (Catalog# PC-49623), shows significantly less potent with CAMKK2 (IC50=27 uM).
PC-49623

SGC-CAMKK2-1

CaMKK2 inhibitor

SGC-CAMKK2-1 is a potent, selective chemical probe inhibitor that targets CaMKK2 with enzyme IC50 of 30 nM.
PC-49436

NCS-382

GHBR inhibitor

NCS-382 is a a gamma-hydroxybutyrate receptor (GHBR) antagonist, brain-penetrating high nanomolar-affinity ligand selective for the CaMKIIα hub domain, possesses antagonistic properties.
PC-49435

Ph-HTBA

CaMKIIα hub ligand

Ph-HTBA is a mid-nanomolar affinity (Ki=78nM), brain permeable ligand of CaMKIIα hub domain binding site.
PC-72972

AS105

CaMKII inhibitor

AS105 (AS-105) is a highly potent, ATP-competitive CaMKII inhibitor, inhibits CaMKIIδ with IC50 of 8 nM, Ki of 3 nM.
PC-72971

GS-680

CaMKII inhibitor

GS-680 (GS680) is a novel selective and ATP-competitive CaMKII inhibitor with biochemical IC50 of 2.3 and 15.9 nM against CaMKIIδ and CaMKIIα, respectively.
PC-72970

RA608

CaMKII inhibitor

RA608 (RA-608) is a potent, selective, ATP-competitive, orally available CaMKII inhibitor, inhibits human CaMKIIδ, CaMKIIɣ, CaMKIIα, and CaMKIIβ with IC50 of 22, 51, 121, and 1135 nM, respectively.
PC-72969

RA306

CaMKII inhibitor

RA306 (RA-306) is a selective, potent, orally active, ATP-competitive CaMKII inhibitor, inhibits CaMKII delta (IC50=15 nM), gamma (IC50=25 nM), and alpha (IC50=61 nM) isoforms.
PC-72949

TIM-063

CaMKK inhibitor

TIM-063 (TIM063) is a potent, selective, ATP-competitive CaMKK inhibitor with Ki of 0.35/0.2 uM for CaMKKα and CaMKKβ, respectively.
PC-72909

CS640

CaMK1D inhibitor

CS640 (CS-640) is a potent, selective CaMK1D inhibitor with nanomolar range at both the enzymatic and cellular levels.
PC-72908

CaMK1D-IN-18

CaMK1D inhibitor

CaMK1D-IN-18 is a potent, selective CaMK1D inhibitor with IC50 of 31 nM, >150-fold greater activity against CaMK1D than all non-CaMK1 kinases.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com