| Cat. No. |
Product Name |
Information |
| PC-72909 |
CS640
CaMK1D inhibitor
|
CS640 (CS-640) is a potent, selective CaMK1D inhibitor with nanomolar range at both the enzymatic and cellular levels. |
| PC-72908 |
CaMK1D-IN-18
CaMK1D inhibitor
|
CaMK1D-IN-18 is a potent, selective CaMK1D inhibitor with IC50 of 31 nM, >150-fold greater activity against CaMK1D than all non-CaMK1 kinases. |
| PC-43468 |
KN-62
CaMK II inhibitor, P2X7 antagonist
|
KN-62 (KN62) is a specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMK II) with Ki of 900 nM for rat brain CaMK II, also is a potent, noncompetitive antagonist of P2X7 receptor with IC50 of 15 nM in HEK293 cells. |
| PC-63352 |
CAMKK2 inhibitor 4t
CAMKK2 inhibitor
|
CAMKK2 inhibitor 4t is a potent, selective, orally available, brain-penetrant CAMKK2 inhibitor with pIC50 of 8.5. |
| PC-45723 |
STO-609
CaMKK inhibitor
|
STO-609 is a selective and cell-permeable inhibitor of CaM-KK, inhibits recombinant CaM-KKα and CaM-KKβ with Ki of 80 and 15 ng/ml. |
| PC-45443 |
CaMKII-IN-1
CaMKII inhibitor
|
CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM. |
| PC-24564 |
KN-93
CaMK II inhibitor
|
KN-93 is a selective, cell-permeable, reversible and competitive inhibitor calmodulin-dependent kinase type II (CaMKII) with Ki of 0.37 uM. |
| PC-24513 |
Evans Blue
CaMKII-α inhibitor
|
Evans Blue is a selective small-molecule inhibitor of CaMKII-alpha (CaMKII-α) with IC50 of 197.1 nM, also is a potent inhibitor of L-glutamate uptake via the membrane bound excitatory amino acid transporter (EAAT). |
| PC-23447 |
TRIB2 inhibitor 1 hydrochloride
TRIB2 inhibitor
|
TRIB2 inhibitor 1 hydrochloride is a small-molecule binder and inhibitor of Tribbles pseudokinase 2 (TRIB2), downregulates TRIB2 levels at micromolar concentration. |
| PC-23446 |
TRIB2 inhibitor 1
TRIB2 inhibitor
|
TRIB2 inhibitor 1 is a small-molecule binder and inhibitor of Tribbles pseudokinase 2 (TRIB2), downregulates TRIB2 levels at micromolar concentration. |
