| Cat. No. |
Product Name |
Information |
| PC-27837 |
(R)-BAK2-66
D3R antagonist
|
(R)-BAK2-66 is a potent, selective dopamine D3 receptor (D3R) antagonist with Ki of 6.9 nM, >100-fold more selective for D3R over D2R. |
| PC-27835 |
BP897 hydrochloride
D3R agonist
|
BP897 hydrochloride (BP 897) is a selective D3 dopamine receptor (D3R) partial agonist with Ki of 0.92 nM and 60 nM for D3R and D2R, reduces cocaine-seeking. |
| PC-27834 |
BP897
D3R agonist
|
BP897 (BP 897) is a selective D3 dopamine receptor (D3R) partial agonist with Ki of 0.92 nM and 60 nM for D3R and D2R, reduces cocaine-seeking. |
| PC-27833 |
(R)-VK4-116
D3R antagonist
|
(R)-VK4-116 is a potent, selective dopamine D3 receptor (D3R) antagonist. |
| PC-27261 |
SD2-2305
DRD2 antagonist
|
SD2-2305 is a potent dopamine receptor D2 (DRD2) antagonist, induces caspase-dependent apoptosis in CRC cells. |
| PC-27156 |
NGD94-1
Dopamine D4 receptor antagonist
|
NGD94-1 (NGD 94-1) is a potent and selective dopamine D4 receptor (D4R) antagonist with Ki of 3.6 nM for cloned human D4.2 receptor. |
| PC-26861 |
PG01037 dihydrochloride
D3R antagonist
|
PG01037 dihydrochloride is a potent selective dopamine D3 receptor (D3R) antagonist with binding Ki of 0.7 nM, displays 133- and 540-fold selectivity over D2 and D4 receptors, respectively. |
| PC-26860 |
PG01042
D3R agonist
|
PG01042 is a high affinity, selective D3 dopamine receptor (D3R) agonist with Ki of 0.47 nM, 39-fold selective over D2R. |
| PC-26137 |
ENX-104
D2/D3 receptor antagonist
|
ENX-104 is a highly selective and potent dopamine D2/D3 receptor antagonist with IC50 of 1.1 nM, 0.1 nM, 2.4 nM and 15.3 nM for D2-like inhibitory dopamine receptors D2S, D2L, D3, and D4 respectively. |
| PC-26129 |
Thioridazine
D2R antagonist
|
Thioridazine is a selective antagonist of dopamine receptor D2 family proteins, exhibits potent anti-psychotic and anti-anxiety activities. |
| PC-26051 |
7-OH-DPAT
D3 dopamine receptor agonist
|
7-OH-DPAT (7-Hydroxy-DPAT) is a selective D3 dopamine receptor (D3R) agonist, exhibits significant pharmacological activity in modulating locomotor behavior and dopamine metabolism within the brain. |
| PC-25355 |
D-583
D2/D3 agonist
|
D-583 is a potent hybrid D2/D3 agonist and iron (II)-specific chelator with EC50 of 3.14 nM (Emax=63%) and 0.62 nM (Emax=68%) for D2 and D3 receptors respectively, exhibits anti-ferroptotic activity. |
