| Cat. No. |
Product Name |
Information |
| PC-21656 |
ERW1041E
TG2 inhibitor
|
ERW1041E is a specific, irreversible small molecule transglutaminase 2 (TGase 2; TG2) inhibitor with Ki of 11 uM. |
| PC-21655 |
MD102
TG2 inhibitor
|
MD102 is a potent transglutaminase 2 (TGase 2; TG2) inhibitor with IC50 of 0.35 uM, shows p53 stabilization effect and anticancer activity at RCC cell lines. |
| PC-38770 |
ZED1227
TG2 inhibitor
|
ZED1227 is a potent, selective, covalent, and orally active transglutaminase 2 (TGase 2, TG2) inhibitor with IC50 of 45 nM. |
| PC-35734 |
TTGM 5826
TGase inhibitor
|
TTGM 5826 (TTGM5826, TTGM-5826) is a small molecule, potential modulator of tissue transglutaminase (tTG) conformation. |
| PC-35603 |
JHU-083
Glutaminase inhibitor
|
JHU-083 is an orally available prodrug of the glutaminase inhibitor 6-diazo-5-oxo-L-norleucine (DON), blocks glutaminase activity in brain CD11b+ cells and prevents depression-associated behaviors induced by chronic social defeat stress.. |
| PC-35093 |
UPGL00004
Glutaminase inhibitor
|
UPGL00004 (UPGL 00004) is a potent, allosteric inhibitor of glutaminase C (GAC) with IC50 of 29 nM. |
| PC-43147 |
BPTES
GLS1 inhibitor
|
BPTES is a potent, selective kidney-type glutaminase 1 (GLS1) inhibitor with Ki of 3 uM (rat KGA), selective for GLS1 over GLS2, glutamate dehydrogenase, and γ-glutamyl transpeptidase. |
| PC-43146 |
Glutaminase C inhibitor 968
Gutaminase C inhibitor
|
Glutaminase C inhibitor 968 is a small molecule allosteric inhibitor of glutaminase C (GAC) catalytic activity with Kd of 3 uM, specifically inhibited the growth of transformed cells and various cancer cells by blocking GAC activation. |
| PC-42986 |
GK921
TG2 inhibitor
|
GK921 is a specific, orally active Transglutaminase 2 (TGase 2, TG2) inhibitor with IC50 of 7.71 uM against recombinant hTGase 2. |
| PC-42933 |
CB-839
Glutaminase inhibitor
|
CB-839 (Telaglenastat) is a potent, selective, and orally bioavailable inhibitor of glutaminase with IC50 of 28 and 23 nM for glutaminase in kidney and brain (GAC and KGA), but not the liver form of glutaminase (GLS2, IC50>1 uM). |
| PC-61055 |
Z-DON
Tissue transglutaminase inhibitor
|
Z-DON (Z-ZON-Val-Pro-Leu-OMe) is a potent, irreversible and cell permeable inhibitor of tissue transglutaminase with IC50 of 20 nM. |
| PC-61053 |
L 682777
hTG2 inhibitor
|
L 682777 is a potent, irreversible inhibitor of human tissue transglutaminase (hTG2). |
