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Cat. No. Product Name Information
PC-61142

AZD-9362

AZD-9362 (AZD9362) is a potent, selective, orally bioavailable IGF-1R inhibitor with IC50 of 14 nM.
PC-60348

BI 885578

BI 885578 (BI-885578, BI885578) is a potent,selective, ATP-competitive IGF1R/InsR tyrosine kinase inhibitor with Kd of 9 nM/12 nM, IC50 of 1 nM/1 nM, respectively.
PC-42487

NVP-ADW742

IGF-1R inhibitor

NVP-ADW742 is a selective IGF-1R kinase inhibitor that with IC50 of 0.17 uM in in cellular autophosphorylation assays.
PC-42436

Linsitinib

IGF-1R inhibitor

Linsitinib (ASP-7487, OSI-906) is a potent, selective, orally active, dual IGF-1R/insulin receptor inhibitor with IC50 of 35/75 nM, respectively.
PC-42636

GSK1904529A

IGF-1R inhibitor

GSK1904529A is a potent, selective, ATP-competitive inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM.
PC-42444

BMS-754807

BMS-754807 (BMS 754807, BMS754807) is a potent, reversible, orally active inhibitor of IGF-1R/Insulin receptor with IC50 of 1.8 and 1.7 nM, respectively.
PC-45879

NVP-AEW541

IGF-1R inhibitor

NVP-AEW541 (AEW-541, AEW541) is a potent, and selective inhibitor of IGF-1R with IC50 of 86 nM.
PC-49759

GTX-134

IGF-1R/IR inhibitor

GTx-134 (GTx 134) is a selective small-molecule inhibitor of IGF-1R and insulin receptor (IR) with biochemical IC50 of 97 nM and 187 nM, respectively.
PC-49233

BM001

GH/IGF1 inhibitor

BM001 (BM-001) is a small molecular inhibitor of the integral growth hormone/insulin‐like growth factor‐1 (GH/IGF1) axis, shows potent antiproliferative effect on cancer cells MDA-MM-231 and Colo-205 with IC50 of 20-30 nM.
PC-62993

BMS 695735

BMS 695735 is a potent, selective IGF-1R inhibitor with IC50 of 34 nM.
PC-61008

WP760

A bis-anthracycline and melanoma selective agent that demonstrates anti-melanoma activity at low nanomolar concentrations.
PC-42488

AG1024

A specific IGF-1R inhibitor that inhibits IGF-1R autophosphorylation with IC50 of 7 uM.

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