| Cat. No. |
Product Name |
Information |
| PC-61743 |
MRS 2179
|
MRS 2179 is a potent, selective, competitive P2Y1 receptor antagonist with Kb of 100 nM. |
| PC-61587 |
Elinogrel
|
Elinogrel (PRT060128) is a selective, reversible, competitive and direct-acting P2Y12 receptor antagonist for the treatment of acute coronary syndrome and prevention of secondary thrombotic events.. |
| PC-61586 |
BX-667
|
BX-667 is a potent P2Y12 receptor antagonist that blocks ADP-induced platelet aggregation in human, dog and rat blood (IC50=97, 317 and 3000 nM respectively). |
| PC-61585 |
Cangrelor tetrasodium
|
Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets. |
| PC-61535 |
SAR-216471 hydrochloride
|
SAR-216471 is a potent, highly selective, intravenous and oral, reversible P2Y12 receptor antagonist with binding IC50 of 17 nM. |
| PC-61413 |
BPTU
|
A potent, highly selective and allosteric antagonist of P2Y1 receptor with Ki of 6 nM for hP2Y1. |
| PC-61411 |
MRS-2500 tetraammonium
|
A highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. |
| PC-61410 |
MRS-2365
|
A highly potent, selective P2Y1 receptor agonist with EC50 of 1.2 nM. |
| PC-46930 |
Suramin
|
An antitrypansomal drug that also possesses antitumor activity. |
| PC-45275 |
Clopidogrel hydrogen sulfate
|
A thienopyridine-class antiplatelet agent that works by irreversibly inhibiting P2Y12 receptor on platelets. |
| PC-44770 |
Clopidogrel thiolactone
|
A thienopyridine-class antiplatelet agent that works by irreversibly inhibiting P2Y12 receptor on platelets. |
| PC-44297 |
Clopidogrel
|
A thienopyridine-class antiplatelet agent that works by irreversibly inhibiting P2Y12 receptor on platelets. |
