| Cat. No. |
Product Name |
Information |
| PC-63545 |
E7046
|
E7046 (Palupiprant, ER-886046) is a potent, selective, orally bioavailable EP4 receptor antagonist with IC50 of 13.5 nM, Ki of 23.14 nM. |
| PC-62041 |
U-46619
TP agonist
|
U-46619 is a potent and stable thromboxane A2 (TP) receptor agonist with EC50 of 35 nM. |
| PC-61565 |
MK-7246
CRTH2/GPR44 inhibitor
|
MK-7246 is a potent, selectie, orally available prostaglandin D2 receptor (CRTH2, GPR44) antagonist with Ki of 2.5 nM (hCRTH2). |
| PC-61563 |
BI 671800
|
BI 671800 is a potent, oral prostaglandin D2 receptor (CRTH2) antagonist for treatment of asthma. |
| PC-60673 |
AM211
|
AM211 (AM-211) is a potent, selective and orally bioavailable prostaglandin D2 receptor type 2 (DP2) antagonist with IC50 of 4.9 nM for human DP2. |
| PC-45075 |
Fevipiprant
|
Fevipiprant (NVP-QAW039, QAW-039) is a potent, selective, slowly dissociating CRTh2 antagonist with Kd of 1.14 nM. |
| PC-42700 |
CJ-042794
EP4 antagonist
|
CJ-042794 (CJ-42794) is a potent, selective prostaglandin E receptor subtype 4 (EP4) antagonist with pKi of 8.5. |
| PC-46004 |
MRE-269
IP receptor inhibitor
|
MRE-269 (ACT-333679) is a potent, selective IP receptor (prostaglandin I2 receptor) agonist with Ki of 20 nM. |
| PC-45896 |
ONO-AE3-208
EP4 antagonist
|
ONO-AE3-208 (AE3-208) is a potent, selective EP4 receptor antagonist with Ki of 1.3 nM. |
| PC-45118 |
Terutroban
|
Terutroban (S-18886) is a potent, selective antagonist of the thromboxane receptor (Prostanoid TP receptor) that blocks thromboxane induced platelet aggregation and vasoconstriction. |
| PC-45579 |
PF-04418948
EP2 antagonist
|
PF-04418948 (PF 04418948) is a novel potent and selective prostaglandin EP2 receptor antagonist. |
| PC-45077 |
Grapiprant
EP4 antagonist
|
Grapiprant (CJ-023423, AAT-007) is a potent, selective EP4 receptor antagonist with Ki values of 13/20 nM against human and rat EP(4) receptors. |
