| Cat. No. |
Product Name |
Information |
| PC-49843 |
1G244
DPP8/9 inhibitor
|
1G244 is a potent and selective DPP8/9 inhibitor with IC50 of 14/53 nM and Ki of 0.9/4.2 nM, respectively. |
| PC-49042 |
MK-0626
DPP-4 inhibitor
|
MK-0626 (MK-626) is a potent, selective and orally active DPP-4 inhibitor (IC50=6.3 nM) with excellent selectivity. |
| PC-72074 |
BR102910
FAP inhibitor
|
BR102910 (BR 102910) is a novel potent, selective, oral fibroblast activation protein (FAP) inhibitor with IC50 of 1 nM. |
| PC-72073 |
BR103354
FAP inhibitor
|
BR103354 (BR 103354) is a novel potent, selective, oral fibroblast activation protein (FAP) inhibitor with IC50 of 14 nM. |
| PC-36075 |
UAMC-1110
FAP inhibitor
|
UAMC-1110 (UAMC1110) is a small molecule inhibitor of fibroblast activation protein (FAP). |
| PC-35918 |
KR-62436
DPP-4 inhibitor
|
KR-62436 (KR62436) is a potent, selective DPP4 inhibitor with IC50 of 0.78, 0.49, 0.14 uM for rat plasma, porcine kidney, human DPP4 (Caco-2), respectively. |
| PC-63358 |
TAK-100
DPP-4 inhibitor
|
TAK-100 is a potent, selective and orally active inhibitor of DPP-4 with IC50 of 5.3 nM, shows no inhibition on DPP2/8/9.. |
| PC-50014 |
Talabostat
DPP4 inhibitor
|
Talabostat (PT-100, Val-boroPro) is a potent, nonselective, orally available inhibitor of post-proline cleaving serine proteases with Ki of 0.18 nM for DPP4, also potently inhibits DPP8/9 (IC50=1.5/0.76 nM), FAP, DPP2 and some other DASH family enzymes. |
| PC-43412 |
Talabostat mesylate
DPP4 inhibitor
|
Talabostat (PT-100, Val-boroPro) is a potent, nonselective, orally available inhibitor of post-proline cleaving serine proteases with Ki of 0.18 nM for DPP4, also potently inhibits DPP8/9 (IC50=1.5/0.76 nM), FAP, DPP2 and some other DASH family enzymes. |
| PC-43097 |
DBPR108
DPP4 inhibitor
|
Prusogliptin (DBPR108) is a potent, selective, orally bioavailable and long-acting inhibitor of DPP4 with IC50 of 15 nM, >3,000-fold selectivity over DPP8, DPP9, FAP and DPP-II. |
| PC-63161 |
AZD-5248
DPP-1 inhibitor
|
AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1). |
| PC-61445 |
Evogliptin
DPP-4 inhibitor
|
Evogliptin (DA1229) is a potent, long acting, reversible and competitive DPP-4 inhibitor with IC50 of 0.9 nM. |
