| Cat. No. |
Product Name |
Information |
| PC-62003 |
Zinterol hydrochloride
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-62002 |
Zinterol
|
Zinterol (MJ 9184) is a potent and selective β2 adrenoceptor agonist with pKb of 8.3, displays >2 logs selectivity over β1 (pKb<5.7). |
| PC-61871 |
PF-00610355
|
PF-00610355 (PF 610355) is a potent, selective, and long-acting β2-adrenoreceptor agonist with EC50 of 0.26 nM. |
| PC-61777 |
Xamoterol
|
Xamoterol (ICI 118587) is a third-generation adrenergic β1 adrenergic receptor partial agonist that acts as a cardiac stimulant.. |
| PC-61776 |
STD-101-D1
|
STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM. |
| PC-61509 |
TAK-259 hydrochloride
|
A potent and selective human α1D adrenoceptor (α1D-AR) antagonist with Ki of 1.1 nM. |
| PC-61508 |
TAK-259
|
A potent and selective human α1D adrenoceptor (α1D-AR) antagonist with Ki of 1.1 nM. |
| PC-70285 |
β2AR-IN-15
|
An allosteric, small-molecule negative modulator for β2AR with Kd of 1.7 uM. |
| PC-60704 |
ARC 239 dihydrochloride
|
A potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors. |
| PC-60703 |
BRL 44408 maleate
|
A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-60702 |
BRL 44408
|
A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors. |
| PC-70210 |
Levosalbutamol
|
A short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructive pulmonary disease (COPD).. |
