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Cat. No. Product Name Information
PC-49015

DLCI-1 dihydrochloride

CYP2A6 inhibitor

DLCI-1 dihydrochloride is a potent and selective CYP2A6 inhibitor with IC50 of 17 nM, 15-765-fold selectivity other major hepatic CYP enzymes.
PC-49014

DLCI-1

CYP2A6 inhibitor

DLCI-1 is a potent and selective CYP2A6 inhibitor with IC50 of 17 nM, 15-765-fold selectivity other major hepatic CYP enzymes.
PC-72686

DX308

CYP26 inhibitor

DX308 is a potent, selective dual CYP26A1/B1 inhibitor and retinoic acid metabolism blocking agent.
PC-72684

DX314

CYP26B1 inhibitor

DX314 is a potent, specific CYP26B1 inhibitor with IC50 of 108 nM, >15-fold selectivity over CYP26A1.
PC-72679

8-BOA

CYP4Z1 inhibitor

8-BOA is a selective and potent mechanism-based inactivator of breast cancer-associated CYP4Z1.
PC-35319

HET0016

CYP4A inhibitor

HET0016 (HET-0016) is a potent, selective inhibitor of CYP4A, potently inhibits the formation of 20-HETE with IC50 of 8.9 nM in human renal microsomes.
PC-42617

Cobicistat

CYP3A inhibitor

Cobicistat (GS-9350) is a pharmacoenhancer that acts as potent and selective inhibitor of human CYP3A with IC50 of 30-285 nM.
PC-21449

Dual CYP19A1/CYP11B2 inhibitor X21

CYP19A1/CYP11B2 inhibitor

Dual CYP19A1/CYP11B2 inhibitor X21 is a potent and selective dual inhibitor of aromatase (CYP19A1) and aldosterone synthase (CYP11B2) with IC50 of 2.3 nM and 29 nM, respectively.
PC-21418

TPP-IOA

Cyt c peroxidase inhibitor

TPP-IOA is a specific inhibitor of cytochrome c (cyt c) peroxidase activity, inhibits peroxidase activity of cardiolipin-induced cytochrome c peroxidase activity with IC50 of 5 uM.
PC-20707

TP0472993

20-HETE synthesis inhibitor

TP0472993 is a potent, selective 20-Hydroxyeicosatetraenoic acid (20-HETE) synthesis inhibitor, inhibits 20-HETE formation in human and rat renal microsomes with IC50 of 29 and 347 nM, respectively.
PC-20618

Decursin

CYP2J2 inhibitor

Decursin ((+)-Decursin) is a potent anti-tumor agent and a potent protein kinase C activator, induces apoptosis and cell cycle arrest at G1 phase.
PC-20617

LKY-047

CYP2J2 inhibitor

LKY-047 (LKY047) is a potent, highly selective and reversible competitive cytochrome P450 CYP2J2 (CYP2J2) inhibitor with IC50 of 1.7 uM.

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