| Cat. No. |
Product Name |
Information |
| PC-43271 |
AZD9496 maleate
|
A potent, selective estrogen receptor downregulator (SERD) with ER downregulation pIC50 of 9.68. |
| PC-43270 |
AZD9496
Estrogen receptor inhibitor
|
AZD9496 is a potent, selective estrogen receptor downregulator (SERD) with ER downregulation pIC50 of 9.68. |
| PC-42580 |
XCT790
|
A potent and selective ERRα inverse agonist with IC50 of 300-500 nM in transient transfection assays. |
| PC-46618 |
Clomiphene citrate
|
A non-steroidal, a widely used fertility agent that inhibits estrogen receptor in the hypothalamus. |
| PC-45541 |
Endoxifen hydrochloride
|
A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.. |
| PC-45540 |
Endoxifen
|
A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.. |
| PC-45096 |
(Z)-4-Hydroxytamoxifen
|
A major metabolite of tamoxifen, a well-known Estrogen receptor antagonist in breast but partial estrogen receptor agonist in endometrium. |
| PC-45768 |
SNG-1153
|
A derivate of icaritin that inhibits the growth of lung CSCs. |
| PC-21730 |
ERB-041
ERβ agonist
|
Prinaberel (ERB-041) is a potent, selective estrogen receptor beta (ERβ) agonist with IC50 of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. |
| PC-21622 |
Fulvestrant
ER inhibitor
|
Fulvestrant (ICI 182780) is a steroidal antiestrogen, and potent, specific estrogen receptor (ER) antagonist with IC50 of 0.94 nM. |
| PC-21173 |
Raloxifene
SERM
|
Raloxifene (Keoxifene, LY139481) is potent, selective estrogen receptor modulator (SERM). |
| PC-20995 |
X15695
ERα degrader
|
X15695 is a potent, selective and orally active estrogen receptor alpha (ERα) degrader, destabilizes ERα and stabilizes p53, inhibits ER+ breast cancer cell growth. |
