Cat. No. |
Product Name |
Information |
PC-45044 |
Nexturastat A
HDAC6 inhibitor
|
Nexturastat A is a potent and selective HDAC6 inhibitor with IC50 of 5 nM. |
PC-45702 |
HPOB
HDAC6 inhibitor
|
HPOB is a potent and selective HDAC6 inhibitor (IC50=56 nM). |
PC-45538 |
HDAC3 inhibitor BG45
HDAC3 inhibitor
|
HDAC3 inhibitor BG45 (BG45) is a potent and selective HDAC3 inhibitor with IC50 of 289 nM, shows selectivity over HDAC1 and HDAC2. |
PC-45462 |
TMP269
class IIa HDAC inhibitor
|
TMP269 (TMP 269) is a potent and selective class IIa HDAC inhibitor with IC50s of 126/80/36/19 nM for HDAC4/5/7/9. |
PC-45089 |
MC1568
class IIa HDAC inhibitor
|
MC1568 is a potent and selective class IIa HDAC inhibitor with IC50 of 220 nM for maize HD1-A. |
PC-42902 |
Entinostat
class I HDAC inhibitor
|
Entinostat (MS275) is a potent and selective class I HDACs inhibitor with IC50 of 243/453/248 nM for HDAC1/2/3. |
PC-45619 |
BML-210
HDAC inhibitor
|
BML-210 is a small molecule histone deacetylase (HDAC) inhibitor that induces Ac-histone in A549 cells with EC50 of 181 uM. |
PC-42249 |
CXD101
class I HDAC inhibitor
|
Zabadinostat (CXD101) is a potent, selective and orally active class I HDAC inhibitor with IC50s of 63 nM, 570 nM and 550 nM for HDAC1, HDAC2 and HDAC3, respectively, has no activity against class II HDACs. |
PC-42671 |
Valproic acid sodium salt
HDAC inhibitor
|
Valproic acid sodium salt is a HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. |
PC-42670 |
Valproic acid
HDAC inhibitor
|
Valproic acid is a HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. |
PC-42421 |
EDO-S101
HDAC inhibitor
|
EDO-S101 (Tinostamustine) is a fusion molecule comprising of the alkylator bendamustine and the HDAC-inhibitor vorinostat. |
PC-42767 |
Abexinostat
HDAC inhibitor
|
PCI-24781 (Abexinostat, CRA 024781) is a broad spectrum HDAC inhibitor, inhibits pure recombinant HDAC1 with Ki of 7 nM. |