| Cat. No. |
Product Name |
Information |
| PC-35577 |
ACT-246475
P2Y12 antagonist
|
ACT-246475 (ACT246475) is a potent, selective, reversible P2Y12 receptor antagonist with binding IC50 of 1.0 nM. |
| PC-35051 |
PPTN trifluoroacetate salt
P2Y14 antagonist
|
PPTN is a potent, highly specific antagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays. |
| PC-35050 |
PPTN
P2Y14 antagonist
|
PPTN is a potent, highly specific antagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays. |
| PC-62046 |
YM-254890
Gq signaling inhibitor
|
YM 254890 is a selective Gq signaling inhibitor that strongly inhibits intracellular calcium ion mobilization and serum response element (SRE)-mediated transcription stimulated by several receptors coupled to Gq, but not those coupled to Gi, Gs, or G15. |
| PC-61584 |
Cangrelor
P2Y12 antagonist
|
Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets. |
| PC-61412 |
MRS-2500
P2Y1 inhibitor
|
MRS-2500 is a highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. |
| PC-42218 |
Ticagrelor
P2Y12 antagonist
|
Ticagrelor (AZD6140) is a potent, selective, reversible and oral P2Y12 receptor antagonist with pKi of 8.7. |
| PC-22103 |
PPTN hydrochloride
P2Y14 antagonist
|
PPTN hydrochloride is a potent, highly specific antagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays. |
| PC-22102 |
PPTN
P2Y14 antagonist
|
PPTN is a potent, highly specific antagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays. |
| PC-21206 |
PSB-0739
P2Y12 antagonist
|
PSB-0739 is a high potent, non-nucleotide-derived competitive antagonist of platelet P2Y12 receptor with Ki of 24.9 nM. |
| PC-20994 |
MRS2768 tetrasodium salt
P2Y2R agonist
|
MRS2768 is a selective P2Y2 receptor agonist with EC50 of 1.89 uM, shows no effect for human P2Y4 or P2Y6 receptors. |
| PC-20993 |
AR-C118925
P2Y2R antagonist
|
AR-C118925 is a potent, selective, competitive P2Y2 receptor antagonist with pA2 values of 37.2 nM and 51.3 nM in calcium and β-arrestin assays, respectively. |
