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Cat. No. Product Name Information
PC-60323

CCR2-RA-[R]

CCR2 antagonist

CCR2-RA-[R] is a potent, selective, allosteric CCR2 antagonist with IC50 of 103 nM.
PC-60322

BMS-681

BMS-687681 (BMS-681) is a potent and orally bioavailable dual antagonist of CCR2 and CCR5 with binding IC50 of 0.7 nM and 2.4 nM, respectively.
PC-60261

Chalcone 4 hydrate

CXCL12 inhibitor

Chalcone 4 hydrate is a potent, selective inhibitor of CXCL12 binding to CXCR4 and CXCR7 with IC50 of 200 nM.
PC-60260

VUF11403

CXCR7 agonist

VUF11403 is a potent CXCR7 (ACKR3) agonist with pKi of 8.1 (hCXCR7), induces recruitment of β-arrestin2 and subsequent internalization of CXCR7.
PC-60259

VUF11207 fumarate

VUF11207 fumarate is a potent CXCR7 (ACKR3) agonist with EC50 of 1.6 nM, inducse recruitment of β-arrestin2 and subsequent internalization of CXCR7 in cells.
PC-60244

(S)-CCX-777

CXCR7 agonist

(S)-CCX-777 is a small-molecule partial agonist of CXCR7 (ACKR3)..
PC-60243

(R)-CCX-777

CXCR7 agonist

(R)-CCX-777 is a small-molecule partial agonist of CXCR7 (ACKR3), the (R)-form of CCX777.
PC-60242

CCX-777

CXCR7 agonist

CCX-777 is a small-molecule partial agonist of CXCR7 (ACKR3).
PC-60240

CCX2553

CCR6 antagonist

CCX2553 is a potent and specific CCR6 antagonist.
PC-60212

CCX-771

CXCR7 inhibitor

CCX-771 is a potent, selective CXCR7 antagonist with IC50 of 4.1 nM.
PC-45710

Danirixin

CXCR2 antagonist

Danirixin (GSK1325756) is a high-affinity, selective and reversible CXCR2 antagonist (IC50=12.5 nM, CXCL8.
PC-47505

Motixafortide

CXCR4 antagonist

Motixafortide (BL-8040, BKT-140, TF-14016) is a 14-residue biostable synthetic peptide, high-affinity CXCR4 antagonist (IC50=1 nM).

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