| Cat. No. |
Product Name |
Information |
| PC-49099 |
5J89LIG
PD-L1 inhibitor
|
5J89LIG is a small molecule h-PD1/h-PD-L1 interaction inhibitor with IC50 of 18.0 nM, bind specifically to hPD-L1 through a unique mode of action, induces the dimerization of hPD-L1. |
| PC-49097 |
BMS135
PD-L1 inhibitor
|
BMS135 is a small molecule h-PD1/h-PD-L1 interaction inhibitor with IC50 of 79.1 nM, bind specifically to hPD-L1 through a unique mode of action, induces the dimerization of hPD-L1. |
| PC-38391 |
Evixapodlin
PD-1/PD-L1 inhibitor
|
Evixapodlin (GS-4224) is a highly potent, small molecule human PD-1/PD-L1 protein-protein interaction inhibitor with IC50 of 0.213 nM, exhibits potential anticancer and antiviral activities. |
| PC-73047 |
PD-L1 inhibitor 4
PD-L1 inhibitor
|
PD-L1 inhibitor 4 is a small molecule inhibitor of PD-1/PD-L1 with SPR KD of 0.079 nM. |
| PC-72848 |
INCB086550
PD-L1 inhibitor
|
INCB086550 (INCB 086550) is a potent, selective small-molecule inhibitor of PD-L1, inhibits PD-L1/PD-1 interaction with IC50 of 3.1, 4.9 and 1.9 nM for human, cynomolgus and rat PD-L1 in HTRF-based assays. |
| PC-72764 |
ZE132
PD-L1 inhibitor
|
ZE132 is a potent and selective small-molecule inhibitor of PD-1/PD-L1 interaction with IC50 of <0.1 nM. |
| PC-72654 |
CA-170
VISTA/PD-L1 inhibitor
|
CA-170 (CA170) is a first-in-class, orally available, tripeptide small-molecule dual antagonist of VISTA/PD-L1, important negative checkpoint regulators of immune activation. |
| PC-35244 |
PD1-PD L1 inhibitor Polaris
|
PD1-PD L1 inhibitor Polaris is a novel potent, small molecule inhibitor of PD-1/PD-L1 interaction (IC50=0.1-10 nM in ELISA assays) with anti-cancer activity. |
| PC-70037 |
BMS-1166 hydrochloride
|
BMS-1166 Hcl salt is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 1.4 nM in a homogenous time-resolved fluorescence binding assay. |
| PC-70036 |
BMS-1166
|
BMS-1166 is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 1.4 nM in a homogenous time-resolved fluorescence binding assay. |
| PC-70035 |
BMS-1001 hydrochloride
|
BMS-1001 is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 2.25 nM in a homogenous time-resolved fluorescence binding assay. |
| PC-70034 |
BMS-1001
|
BMS-1001 is a potent PD-1/PD-L1 interaction inhibitor with IC50 of 2.25 nM in a homogenous time-resolved fluorescence binding assay.. |
