Cat. No. |
Product Name |
Information |
PC-72325 |
MS910
MEK1/2 degrader
|
MS910 (MS-910) is the first CRBN-recruiting MEK1/2 degrader (PROTC) with HT29 DC50 of 118/55 nM for MEK1/2 degradation, respectively. |
PC-72324 |
MS934
MEK1/2 degrader
|
MS934 (MS-934) is a VHL-recruiting MEK1/2 degrader (PROTAC) with HT29 DC50 of 18/9 nM for MEK1/2 degradation, respectively. |
PC-72322 |
dBRD9‐A
BRD9 degrader
|
dBRD9‐A is a chemical degrader (PROTAC) of BRD9, a highly specific binder of the BRD9 bromodomain and elicits near complete BRD9 degradation at low nanomolar concentrations. |
PC-72286 |
MS177
EZH2 PROTAC
|
MS177 (MS-177) is a potent and selective EZH2 degarder (PROTAC) based on EZH2 inhibitor C24 with CRBN ligand pomalidomide with DC50 of 0.2 uM in EOL-1 cells. |
PC-72115 |
CG428
Trk degrader
|
CG428 (CG-428) is a first-in-class potent and selective TRK degrader (PROTAC) with DC50 of 0.36 nM. |