| Cat. No. |
Product Name |
Information |
| PC-45789 |
Clemizole
|
An H1 histamine receptor antagonist that substantially inhibits HCV replication by suppression of NS4B's RNA binding (IC50=24 nM) with little toxicity for the host cells. |
| PC-42591 |
Capsaicin
|
An active component of chili pepper, potent agonist of TRPV1 channel with EC50 of 0.29 uM.. |
| PC-45042 |
SN-2
|
A small molecule activator of the TRPML3 ion channel with EC50 of 1.13 uM. |
| PC-42062 |
JNJ-17203212
|
A potent, selective and orally bioavailable TRPV1 receptor antagonist with IC50 of 65 nM and 102 nM for hTRPV1 and rTRPV1, respectively. |
| PC-42688 |
SB-705498
|
A potent, selective and orally bioavailable TRPV1 antagonist with pKi of 7.6 (inhibition of capsaicin-mediated activation of hTRPV1 receptor). |
| PC-45556 |
PF-4840154
|
A potent, selective agonist of the rat (EC50=97 nM) and human (EC50=23 nM) TRPA1 channel. |
| PC-42689 |
AMG 517
|
A potent and selective vanilloid receptor TRPV1 antagonist with IC50 of 0.76 nM for hTRPV1. |
| PC-42931 |
SB-366791
|
A potent and selective vanilloid receptor (VR1/TRPV1) antagonist. |
| PC-45764 |
BCTC
|
A highly potent, selective, CNS-penetrant TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 with IC50 values of 35 and 6 nM, respectively. |
| PC-45355 |
Nonivamide
|
A capsaicin analog that acts as an agonist of TRPV1 channel. |
