| Cat. No. |
Product Name |
Information |
| PC-20325 |
HTL0041178
GPR52 agonist
|
HTL0041178 is a potent GPR52 agonist with EC50 of 27.5 nM (human or rat GPR52). |
| PC-20321 |
BC-K-YH16899
KRS-67LR inhibitor
|
BC-K-YH16899 (YH16899) is a specific small molecule inhibitor of prometastatic lysyl-tRNA synthetase-laminin receptor interaction (KRS-67LR PPI), suppresses cancer metastasis. |
| PC-20318 |
Secdin
ARF-GEF inhibitor
|
Secdin is a small-molecule inhibitor of Arabidopsis thaliana ADP-ribosylation factor (ARF)-guanine nucleotide exchange factors (GEFs), impaires both hypocotyl and root growth in young Arabidopsis seedlings with IC50 of 4 uM. |
| PC-20313 |
SJ572946
BAK activator
|
SJ572946 is a small molecule BAK activator, binds to the activation groove of BAK and selectively triggers BAK activation over that of BAX in liposome and mitochondrial permeabilization assays. |
| PC-20305 |
ELOVL6 inhibitor 37
ELOVL6 inhibitor
|
ELOVL6 inhibitor 37 is a potent, selective inhibitor of elongase of long-chain fatty acids family 6 (ELOVL6) with IC50 of 8.9 and 31 nM for human and mouse ELOVL6, respectively. |
| PC-20304 |
ELOVL6 inhibitor Compound A
ELOVL6 inhibitor
|
ELOVL6 inhibitor Compound-A is a potent, selective inhibitor of elongase of long-chain fatty acids family 6 (ELOVL6) with IC50 of 169 and 350 nM for human and mouse ELOVL6, respectively. |
| PC-20302 |
HTS13286
AQP9 inhibitor
|
HTS13286 is a selective AQP9 inhibitor with IC50 of 1.5 uM (inhibition of CHO-AQP9 cell water permeability). |
| PC-20301 |
RF03176
AQP9 inhibitor
|
RF03176 is a selective AQP9 inhibitor with IC50 of 1.3 uM (inhibition of CHO-AQP9 cell water permeability). |
| PC-20300 |
TGN-020
AQP4 inhibitor
|
TGN-020 (TGN020) is a potent, selective aquaporin 4 (AQP4) inhibitor with IC50 of 3 uM. |
| PC-20274 |
SPT inhibitor compound-2
SPT inhibitor
|
SPT inhibitor compound-2 is a potent, orally active serine palmitoyltransferase (SPT) inhibitor with IXC50 of 0.51 nM in cell-free assays. |
| PC-20224 |
Compound 30666
IgH gene enhancer inhibitor
|
Compound 30666 is a specific small molecule inhibitor of IgH enhancer transcriptional activity with IC50 of 2.1 uM, inhibits immunoglobulin production by MM cells. |
| PC-20213 |
2,5-pyridinedicarboxylic acid
MIF2 inhibitor
|
2,5-pyridinedicarboxylic acid is a highly selective D-dopachrome tautomerase (D-DT, MIF2) inhibitor with Ki of 17.2 uM, 79-fold selectivity over MIF, effectively blocks the D-DT-induced activation of CD74. |
