| Cat. No. |
Product Name |
Information |
| PC-20846 |
CC-410
NNMT inhibitor
|
CC-410 (CC410) is a potent, specific inhibitor of nicotinamide N-methyltransferase (NNMT) with IC50 of 1.6 uM (human NNMT). |
| PC-20842 |
GCN2iA
GCN2 inhibitor
|
GCN2iA is a potent seletive inhibitor of general control nonderepressible 2 (GCN2) with IC50 of 4.0 nM. |
| PC-20837 |
SRP-001
Analgesic agent
|
SRP-001 is a non-opioid and non-hepatotoxic small molecule ApAP analog, induces analgesia via N-arachidonoylphenolamine (AM404) formation, and generates higher amounts of AM404 than ApAP. |
| PC-20828 |
LAG-3 inhibitor SA-15-P
LAG-3 inhibitor
|
LAG-3 inhibitor SA-15-P is a small molecule dual inhibitor of LAG-3/MHCII and LAG-3/FGL1 interactions with IC50 of 4.21 and 6.52 uM, respectively. |
| PC-20827 |
DFTD
eEF-2K inhibitor
|
DFTD is a time-dependent, reversible and covalent inhibitor of eukaryotic elongation factor 2 kinase (eEF-2K) targeting of Cys-146, DFTD binds to the ATP binding site of eEF-2K. |
| PC-20825 |
eEF-2K inhibitor 2C
eEF-2K inhibitor
|
eEF-2K inhibitor 2C (Compound 2C) is a small molecule inhibitor of eukaryotic elongation factor 2 kinase (eEF-2K), binds to the ATP-binding site of eEF-2K. |
| PC-20821 |
PKA inhibitor H89
PKA inhibitor
|
PKA inhibitor H89 (H-89 dihydrochloride) is a potent, selective cAMP-dependent protein kinase A (PKA) inhibitor with IC50 of 48 nM, weakly inhibits PKG, PKC, casein kinases. |
| PC-20814 |
Legumain inhibitor 7r
Legumain inhibitor
|
Legumain inhibitor 7r is a highly potent Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 0.9 nM. |
| PC-20813 |
Legumain inhibitor 10t
Legumain inhibitor
|
Legumain inhibitor 10t is a potent, selective and cellularly active Legumain (asparagine endopeptidase, AEP) inhibitor with IC50 of 71 nM. |
| PC-20812 |
Legumain inhibitor 38u
Legumain inhibitor
|
Legumain inhibitor 38u is a selective inhibitor of asparagine endopeptidase (AEP, Legumain) with IC50 of 160 nM, inhibits cancer metastasis. |
| PC-20808 |
L524-0366
FN14 inhibitor
|
L524-0366 is a small-molecule inhibitor of Fn14, binds specifically to the Fn14 receptor and disrupts TWEAK-Fn14 interaction. |
| PC-20806 |
NSC33353
|
NSC33353 (NSC 33353) is a small molecule inhibitor with potent anti-tumor activity against TNBC cells, enhances TNBC sensitivity to doxorubicin. |
